描述
Tizanidine Hydrochloride is an ?2-adrenergic receptor agonist commonly used in laboratory models of muscle spasticity, neuroinhibition, and CNS signaling. Its mechanism involves reducing presynaptic excitatory neurotransmitter release, making it useful in research involving:
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Spinal cord injury
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Neuromuscular dysfunction
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Central inhibition and sedation studies
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Comparative pharmacodynamics with baclofen and diazepam
This product is intended for in vitro and animal research only and is not suitable for therapeutic or diagnostic applications.
Side Effects (Observed in Research Models)
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Drowsiness
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Hypotension
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Dry mouth
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Dizziness
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Bradycardia (at high doses)
Handle with care under institutional safety guidelines.
Product Specifications
Parameter | Details |
---|---|
Product Name | Tizanidine Hydrochloride Tablets (Kailaitong / ???) |
Active Ingredient | Tizanidine Hydrochloride |
CAS Number | 64461-82-1 |
Molecular Formula | C?H?ClN?S·HCl |
Molecular Weight | 290.2 g/mol |
Strength | 2?mg per tablet |
Formulation | Oral tablet |
Quantity per Box | 36 tablets (12 tablets × 3 blister packs) |
Dosage Form | Tablet |
Approval Number | ????H20060645 |
Product Code | 86902181000261 |
Manufacturer | Sichuan Keruide Pharmaceutical Co., Ltd. |
Barcode | 6939234900203 |
Storage Conditions | Store below 25?°C in a dry, sealed environment |
Intended Use | Laboratory research only |
Mechanism of Action
Tizanidine is a centrally acting ?2-adrenergic receptor agonist that inhibits motor neuron activity by suppressing excitatory neurotransmitter release. Its selective action allows for precise modeling of neuromuscular conditions, spasticity control, and sedative interactions in CNS research.
Research Applications
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Muscle spasm and spasticity models
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CNS inhibition and sedation studies
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Neuropharmacological receptor modulation
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Spinal cord injury recovery models
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?2-adrenergic pharmacodynamics
Core Keywords
Tizanidine hydrochloride tablets, CAS 64461-82-1, CNS research tizanidine, alpha-2 agonist lab use, spasticity model drug, tizanidine 2mg Kailaitong, muscle relaxant research, non-clinical tizanidine, wholesale lab-grade tizanidine, neuroinhibitory agent
Research Use Disclaimer
This product is intended strictly for laboratory research purposes. It is not approved for human, diagnostic, clinical, or veterinary use. Proper biosafety and handling procedures should be followed in compliance with institutional protocols.
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