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Lappaconitine Hydrobromide 4?mg ×?2 Ampoules Wholesale price comparison
$3.00
Lappaconitine hydrobromide is a naturally derived diterpenoid alkaloid from Aconitum species, known for analgesic, anti-inflammatory, anti-arrhythmic, and antitumor effects. Each box contains two 2?mL ampoules at 4?mg each. Produced by Shandong Dongfangming Pharmaceutical Group Co., Ltd., NMPA approval number H20045497, product code 86904083001063, barcode 6935030530552.
?? For laboratory research use only.?Please consult the staff for other purposes?
CAS number: 97792?45?5
Description
Product Specifications
| Attribute | Details |
|---|---|
| Product Name | Lappaconitine Hydrobromide Injection |
| Generic Name | Lappaconitine Hydrobromide |
| CAS Number | 97792?45?5 |
| Molecular Formula | C??H??BrN?O? · HBr |
| Molecular Weight | ~665.6?g/mol |
| Dosage Form | Sterile injectable solution |
| Strength | 2?mg/mL (4?mg per 2?mL ampoule) |
| Pack Size | 2 ampoules per box |
| Approval Number | H20045497 (China NMPA) |
| Product Code | 86904083001063 |
| Manufacturer | Shandong Dongfangming Pharmaceutical Group Co., Ltd. |
| Barcode | 6935030530552 |
| Storage | Store at 2–8?°C; light protection |
| Intended Use | Laboratory research use only |
Mechanism of Action
Lappaconitine acts primarily as a voltage-gated sodium channel blocker, inhibiting neuronal signal transmission. It also exhibits anti-arrhythmic activity by blocking cardiac sodium channels and demonstrates additional anti-inflammatory and antitumor effects in vitro and in vivo plantgrowthhormones.com+15drugs.ncats.io+15pmc.ncbi.nlm.nih.gov+15.
Research Applications & Pharmacology
Analgesia models: Effective in treating cancer pain, neuralgia, and postoperative pain without opioids.
Anti-inflammatory studies: Exhibits potent activity in models of inflammation.
Cardiac electrophysiology models: Class I antiarrhythmic effects studied in atrial fibrillation, ventricular arrhythmias.
Pharmacokinetics: Organ-independent metabolism; LD?? in rodents is ~20–32?mg/kg; note narrow therapeutic margin.
Safety Profile & Handling
Observed effects:
Analgesia, anti-inflammatory, and antiarrhythmic responses.
Toxicity includes cardiac and neurological effects; narrow therapeutic window. Monitor closely in animal studies .
Handling precautions:
Use full PPE (gloves, goggles, lab coat).
Prepare in a fume hood; inject IV only.
Dispose of unused ampoules and materials as hazardous chemical waste.
?? Research?Use Disclaimer
This product is intended exclusively for laboratory research. It is not approved for therapeutic, diagnostic, clinical, or veterinary use. Misuse may pose significant risks and compromise research integrity.
Additional information
| Weight | 1.1 kg |
|---|---|
| Dimensions | 18 × 16 × 18 cm |
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